SCHEMBL6972848

SCHEMBL6972848

CC(C)c1nc(CN)n(Cc2cccnc2)c1Sc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.38
ALOX5AP P20292 1/20 0.37
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 1/20 0.36
SRC P12931 1/20 0.34
BLM P54132 1/20 0.34
GABRA1 P14867 2/20 0.34
GABRA5 P31644 2/20 0.34
PKM P14618 1/20 0.34
GNRHR P30968 1/20 0.34
TP53 P04637 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087890 0.92 TLR7 (0.41) TLR7ALOX5APALDH1A1MAPK1SRC
SCHEMBL7081083 0.89 ALOX5AP (0.37) TLR7ALOX5APALDH1A1MAPK1SRC
SCHEMBL6974887 0.88 GRIN1 (0.39) TLR7ALDH1A1SRCCYP3A4CYP2D6
SCHEMBL6965787 0.88 ALDH1A1 (0.38) ALDH1A1SRCGABRA1GABRA5PKM
SCHEMBL6972815 0.88 KDM4E (0.36) TLR7ALOX5APALDH1A1CYP3A4CYP2D6
SCHEMBL6957238 0.88 GABRA5 (0.36) TLR7ALOX5APALDH1A1MAPK1SRC
SCHEMBL7084611 0.88 GRIN1 (0.39) TLR7ALOX5APALDH1A1SRC
SCHEMBL6969489 0.88 ALDH1A1 (0.37) TLR7ALOX5APALDH1A1MAPK1SRC
SCHEMBL7083103 0.87 ALOX5AP (0.36) TLR7ALOX5APALDH1A1MAPK1SRC
SCHEMBL7085922 0.87 CHRNB2 (0.42) TLR7ALOX5APALDH1A1MAPK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed