SCHEMBL6970043

SCHEMBL6970043

N#Cc1cc(CC=O)ccc1-c1ccco1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.41
ALDH1A1 P00352 9/20 0.41
MEN1 O00255 9/20 0.41
KMT2A Q03164 9/20 0.41
HPGD P15428 5/20 0.41
MAPT P10636 5/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
MAPK1 P28482 3/20 0.39
ADORA2A P29274 4/20 0.39
ADORA2B P29275 3/20 0.39
ADORA1 P30542 3/20 0.39
POLB P06746 4/20 0.38
HSD17B10 Q99714 4/20 0.38
BLM P54132 3/20 0.38
GAA P10253 3/20 0.38
ALOX15 P16050 2/20 0.38
USP2 O75604 1/20 0.38
ESR1 P03372 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967431 0.77 MAPT (0.37) KDM4EALDH1A1HPGDMAPTMAPK1
SCHEMBL6963441 0.74 PTPN1 (0.57) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL3567606 0.74 ESR1 (0.51) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL6970040 0.71 KDM4E (0.42) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL6959707 0.71 CFTR (0.49) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL8476284 0.71 MEN1 (0.50) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL31264118 0.71 MEN1 (0.50) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL15196773 0.68 TSHR (0.41) KDM4EALDH1A1TSHR
SCHEMBL4549089 0.68 VCAM1 (0.46) BLM
SCHEMBL2975866 0.68 TRPV4 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649636-B1 Cyclooxygenase inhibitors PFIZER INC. 2003-11-18 US disclosed
EP-1104759-B1 Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents PFIZER PROD INC (US) 2003-10-22 EP disclosed
EP-1104759-A1 Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents Pfizer Products Inc. (US) 2001-06-06 EP disclosed