SCHEMBL6970428

SCHEMBL6970428

CN(C)CCCN1C(=O)CN(C(=O)c2ccc(N)cc2)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.43
LMNA P02545 4/20 0.43
HTR1A P08908 4/20 0.43
DRD2 P14416 4/20 0.43
SLC6A4 P31645 4/20 0.43
CYP1A2 P05177 4/20 0.43
PRNP P04156 3/20 0.43
CHRM2 P08172 3/20 0.43
CHRM1 P11229 3/20 0.43
DRD1 P21728 3/20 0.43
SLC6A2 P23975 3/20 0.43
ADRA1A P35348 3/20 0.43
OPRM1 P35372 3/20 0.43
DRD3 P35462 3/20 0.43
KCNH2 Q12809 3/20 0.43
TSHR P16473 3/20 0.43
SLC6A3 Q01959 2/20 0.43
ADRA2A P08913 2/20 0.43
TBXA2R P21731 1/20 0.43
MAPT P10636 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959648 0.93 AVPR1A (0.42) LMNAHTR1ADRD2SLC6A4CHRM2
SCHEMBL6969600 0.89 AVPR2 (0.46) CYP2D6LMNAHTR1ADRD2SLC6A4
SCHEMBL6969043 0.85 DRD3 (0.47) CYP2D6LMNAHTR1ADRD2SLC6A4
SCHEMBL6970673 0.82 AVPR2 (0.48) LMNAHTR1ADRD2SLC6A4CHRM2
SCHEMBL6967996 0.81 AVPR2 (0.47) HTR1ADRD2SLC6A4CHRM2CHRM1
SCHEMBL6972375 0.78 KDM4E (0.43) LMNAHTR1ADRD2SLC6A4CHRM2
SCHEMBL6959966 0.78 AVPR2 (0.58) AVPR2AVPR1A
SCHEMBL6972489 0.76 AVPR2 (0.63) AVPR2AVPR1A
SCHEMBL27362645 0.75 AVPR2 (0.40) CYP2D6LMNAHTR1ADRD2SLC6A4
SCHEMBL6958687 0.75 DRD3 (0.46) CYP2D6LMNAHTR1ADRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed