SCHEMBL6969043

SCHEMBL6969043

CN(C)CCCN1C(=O)CN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.47
CHRM2 P08172 3/20 0.47
HTR1A P08908 3/20 0.47
DRD1 P21728 3/20 0.47
SLC6A4 P31645 3/20 0.47
ADRA2A P08913 2/20 0.47
PTGS1 P23219 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
BCHE P06276 1/20 0.41
P2RX4 Q99571 1/20 0.41
DRD2 P14416 3/20 0.40
DRD4 P21917 2/20 0.40
CYP2D6 P10635 4/20 0.40
LMNA P02545 2/20 0.40
PRNP P04156 2/20 0.40
CHRM1 P11229 2/20 0.40
SLC6A2 P23975 2/20 0.40
ADRA1A P35348 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972375 0.94 KDM4E (0.43) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL6958687 0.90 DRD3 (0.46) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL6970428 0.85 CYP2D6 (0.43) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL6955542 0.84 ALDH1A1 (0.43) DRD3L3MBTL1ALDH1A1MAPTBCHE
SCHEMBL6964416 0.83 DRD2 (0.50) DRD3HTR1AL3MBTL1ALDH1A1DRD2
SCHEMBL6959648 0.78 AVPR1A (0.42) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL27361135 0.77 XIAP (0.41) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL6959376 0.77 HDAC1 (0.46) HTR1AL3MBTL1ALDH1A1MAPTBCHE
SCHEMBL6969600 0.75 AVPR2 (0.46) DRD3CHRM2HTR1ADRD1SLC6A4
SCHEMBL6971119 0.75 DRD2 (0.46) DRD3L3MBTL1ALDH1A1MAPTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed