SCHEMBL6972183

SCHEMBL6972183

NC(CCc1ccc(CCc2c[nH]cn2)cc1)=NCc1ccc(Cl)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.47
GRIN1 Q05586 2/20 0.47
TAAR1 Q96RJ0 2/20 0.40
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
HRH3 Q9Y5N1 7/20 0.38
HRH4 Q9H3N8 3/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MALT1 Q9UDY8 1/20 0.35
ATP4A P20648 1/20 0.34
ATP4B P51164 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968578 0.92 GRIN2B (0.46) GRIN2BGRIN1TAAR1HTR3EHTR3B
SCHEMBL6974030 0.90 TAAR1 (0.40) GRIN2BGRIN1TAAR1HTR3EHTR3B
SCHEMBL6968091 0.85 GRIN2B (0.53) GRIN2BGRIN1TAAR1HTR3EHTR3B
SCHEMBL224352 0.81 DAO (0.41) TAAR1
SCHEMBL6972175 0.79 TAAR1 (0.40) GRIN2BGRIN1TAAR1HTR3EHTR3B
SCHEMBL6973473 0.74 GRIN2B (0.39) GRIN2BGRIN1TAAR1HTR3EHTR3B
SCHEMBL6955812 0.74 GRIN2B (0.55) GRIN2BGRIN1TAAR1MALT1
SCHEMBL9034160 0.73 MAOB (0.40) TAAR1
SCHEMBL6972503 0.73 MEN1 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9079252 0.73 PLAAT3 (0.40) CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729459-B1 PHENYL-ALKYL IMIDAZOLES AS H3-RECEPTOR ANTAGONISTS SCHERING CORP (US) 2003-03-12 EP disclosed
US-5578616-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, TREATMENT FOR GASTROINTESTINAL AND CARDIOVASCULAR DISORDERS SCHERING CORPORATION (US) 1996-11-26 US disclosed