SCHEMBL6972366

SCHEMBL6972366

CC(C)c1nc(C(Cc2cccnc2)OCCO)[nH]c1Sc1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
IDO1 P14902 1/20 0.32
NPC1 O15118 1/20 0.31
PLA2G7 Q13093 1/20 0.31
GRM5 P41594 1/20 0.30
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
CTSS P25774 1/20 0.30
ADRB2 P07550 1/20 0.30
ADRB1 P08588 1/20 0.30
ADRB3 P13945 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085227 0.93 IDO1 (0.31) KMT2AIDO1
SCHEMBL7084598 0.91 ADRB2 (0.33) ADRB2ADRB1ADRB3
SCHEMBL6962106 0.90 TP53 (0.32) ALDH1A1LMNARAB9AKMT2AIDO1
SCHEMBL7084647 0.90 ALDH1A1 (0.38) ALDH1A1LMNARAB9AKMT2AIDO1
SCHEMBL7085468 0.89 CHRM1 (0.32) LMNAKMT2A
SCHEMBL6967430 0.87 ALDH1A1 (0.41) ALDH1A1LMNARAB9AKMT2AIDO1
SCHEMBL6974934 0.86 CYP19A1 (0.35) ALDH1A1LMNARAB9AKMT2A
SCHEMBL6973902 0.86 IDO1 (0.32) IDO1
SCHEMBL6970038 0.86 ALDH1A1 (0.41) ALDH1A1LMNARAB9AKMT2AIDO1
SCHEMBL7087608 0.85 TP53 (0.35) ALDH1A1GRM5ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed