SCHEMBL7084598

SCHEMBL7084598

CC(C)c1nc(C(Cc2ccncc2)OCCO)[nH]c1Sc1cccc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
PDE4D Q08499 1/20 0.31
PDE4B Q07343 1/20 0.31
SLC6A9 P48067 1/20 0.30
CSNK2A2 P19784 1/20 0.30
CSNK2B P67870 1/20 0.30
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970653 0.92
SCHEMBL6972366 0.91 ALDH1A1 (0.37) ADRB2ADRB1ADRB3
SCHEMBL8799715 0.90 PDE4D (0.32) PDE4DPDE4B
SCHEMBL7084286 0.89 MAPK13 (0.30)
SCHEMBL6973004 0.89 SLC6A9 (0.32) SLC6A9CSNK2A2CSNK2BFNTAFNTB
SCHEMBL6967066 0.89 CYP3A4 (0.32)
SCHEMBL7087608 0.87 TP53 (0.35) ADRB2ADRB1ADRB3SLC6A9
SCHEMBL7081545 0.86 CSNK2A2 (0.34) PDE4DPDE4BSLC6A9CSNK2A2CSNK2B
SCHEMBL6960274 0.86 MAPT (0.34) ADRB2ADRB1ADRB3SLC6A9
SCHEMBL7080474 0.86 CSNK2A2 (0.34) ADRB2ADRB1ADRB3PDE4DPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed