SCHEMBL6972815

SCHEMBL6972815

CC(C)c1nc(CN)n(Cc2ccncc2)c1Sc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
TLR7 Q9NYK1 5/20 0.35
ALOX5AP P20292 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2D6 P10635 1/20 0.33
HIF1A Q16665 1/20 0.33
GSK3B P49841 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNK13 Q9HB14 2/20 0.32
GAA P10253 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082836 0.91 TLR7 (0.38) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL7078348 0.88 SMN1; SMN2 (0.36) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL6967360 0.88 IDO1 (0.36) KDM4EALDH1A1TDP1PIM1PIM3
SCHEMBL6972848 0.88 TLR7 (0.38) KDM4ETLR7ALOX5APALDH1A1CYP3A4
SCHEMBL6971599 0.87 GRIN1 (0.36) KDM4ECYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6967507 0.87 PIM1 (0.34) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL6967403 0.86 GSK3B (0.36) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL6975575 0.86 KDM4E (0.34) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL6960328 0.86 ALDH1A1 (0.37) KDM4ETLR7ALOX5APALDH1A1MAPT
SCHEMBL6957548 0.86 KCNH2 (0.35) TDP1PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed