SCHEMBL7082836

SCHEMBL7082836

CC(C)c1nc(CCN)n(Cc2ccncc2)c1Sc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.38
GSK3B P49841 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
HTR2C P28335 1/20 0.34
HTR6 P50406 1/20 0.34
ALOX5AP P20292 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
ENPP2 Q13822 2/20 0.32
TRPC5 Q9UL62 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972815 0.91 KDM4E (0.36) TLR7GSK3BCYP1A2CYP3A4CYP2D6
SCHEMBL6967403 0.89 GSK3B (0.36) TLR7GSK3BCYP1A2CYP3A4CYP2D6
SCHEMBL6974232 0.89 IDO1 (0.35) TLR7GSK3BKDM4EHTR2CHTR6
SCHEMBL7087890 0.88 TLR7 (0.41) TLR7HIF1AHTR2CHTR6ALOX5AP
SCHEMBL6975055 0.88 GRIN1 (0.35) TLR7GSK3BCYP3A4HTR2CHTR6
SCHEMBL7082703 0.87 KCNH2 (0.34) TLR7GSK3BLOXL2TDP1
SCHEMBL7086620 0.87 GSK3B (0.40) TLR7GSK3BCYP1A2CYP3A4CYP2D6
SCHEMBL7078348 0.86 SMN1; SMN2 (0.36) TLR7GSK3BCYP1A2CYP3A4CYP2D6
SCHEMBL6974036 0.86 ENPP2 (0.33) TLR7GSK3BLOXL2ENPP2
SCHEMBL8347165 0.86 LMNA (0.45) GSK3BENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed