SCHEMBL6972963

SCHEMBL6972963

CC(C)c1nc(CCCOCc2ccccc2)n(Cc2ccncc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.38
TDP1 Q9NUW8 1/20 0.35
TLR7 Q9NYK1 7/20 0.35
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
REN P00797 1/20 0.31
PDE4A P27815 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084679 0.95 TDP1 (0.36) GSK3BTDP1TLR7KDM4E
SCHEMBL5853114 0.90 TDP1 (0.37) GSK3BTDP1TLR7KDM4E
SCHEMBL6974348 0.89 GSK3B (0.34) GSK3BTDP1TLR7HRH4HRH3
SCHEMBL6960981 0.87 TLR8 (0.33) TDP1TLR7HRH4HRH3
SCHEMBL14459814 0.85 TLR7 (0.33) TLR7
SCHEMBL6975492 0.85 HRH4 (0.35) GSK3BTDP1HRH4HRH3
SCHEMBL14439828 0.85 TDP1 (0.40) TDP1
SCHEMBL8349607 0.83 TDP1 (0.32) TDP1TLR7
SCHEMBL6966489 0.83 TLR8 (0.35) GSK3BTDP1TLR7
SCHEMBL6972834 0.83 TLR8 (0.35) TDP1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed