SCHEMBL7084679

SCHEMBL7084679

CC(C)c1nc(CCOCc2ccccc2)n(Cc2ccncc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
GSK3B P49841 3/20 0.35
TLR7 Q9NYK1 4/20 0.32
KDM4E B2RXH2 1/20 0.31
IDO1 P14902 1/20 0.31
TRPC5 Q9UL62 1/20 0.31
MAPT P10636 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31
TP53 P04637 1/20 0.31
RECQL P46063 1/20 0.30
KCNH2 Q12809 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972963 0.95 GSK3B (0.38) TDP1GSK3BTLR7KDM4E
SCHEMBL5853114 0.92 TDP1 (0.37) TDP1GSK3BTLR7KDM4EIDO1
SCHEMBL8349607 0.89 TDP1 (0.32) TDP1TLR7TRPC5
SCHEMBL14439828 0.86 TDP1 (0.40) TDP1MAPTTP53RECQL
SCHEMBL6969339 0.86 ALDH1A1 (0.36) TDP1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6974526 0.86 TDP1 (0.32) TDP1TLR7ALDH1A1
SCHEMBL6973218 0.85 CCR2 (0.41) TDP1KDM4EMAPTCYP2D6CYP2C9
SCHEMBL6964734 0.85 TDP1 (0.33) TDP1ALDH1A1
SCHEMBL6970649 0.84 KCNH2 (0.32) KCNH2
SCHEMBL6974348 0.83 GSK3B (0.34) TDP1GSK3BTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed