Benzofuran

Benzofuran

SCHEMBL6973046

COC(=O)CCc1ccc2c(CC(NC(=O)OCc3ccccc3)C(=O)O)occ2c1.c1ccc2occc2c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 4/20 0.47
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
TYR P14679 1/20 0.41
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
ITGB3 P05106 8/20 0.39
ITGA2B P08514 7/20 0.39
F2 P00734 1/20 0.38
ITGAV P06756 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967105 0.94 CASP1 (0.50) CASP1CTSLCTSBCTSSTYR
SCHEMBL7231340 0.85 CASP1 (0.47) CASP1CTSLCTSBCTSSTYR
Benzofuran SCHEMBL6973042 0.85 CASP1 (0.48) CASP1CTSLCTSBCTSSTYR
SCHEMBL7394442 0.79 TYR (0.52) CASP1CTSLCTSBCTSSTYR
SCHEMBL6967103 0.78 CASP1 (0.51) CASP1CTSLCTSBCTSSTYR
SCHEMBL6964135 0.75 ITGB3 (0.59) ITGB3ITGA2BITGAV
SCHEMBL6973856 0.71 CA12 (0.37) CTSBCTSSITGA4ITGB7ITGB3
SCHEMBL6978547 0.70 ALDH1A1 (0.52) ITGB3ITGA2BALDH1A1
SCHEMBL7231335 0.69 CASP1 (0.47) CASP1CTSLCTSBCTSSITGB3
SCHEMBL22764775 0.69 CTSB (0.72) CASP1CTSLCTSBCTSSITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133491-B1 NOVEL BENZOFURANE DERIVATIVES, PREPARATION METHOD, USE AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AVENTIS PHARMA SA (FR) 2003-02-19 EP disclosed