SCHEMBL6973102

SCHEMBL6973102

CC(C)c1nc(CNS(C)(=O)=O)n(Cc2ccncc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
GNRHR P30968 4/20 0.35
NAMPT P43490 1/20 0.32
TP53 P04637 2/20 0.31
MAPT P10636 1/20 0.31
POLB P06746 1/20 0.31
THRB P10828 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ENPP2 Q13822 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP21A2 P08686 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967611 0.92 GRIN1 (0.35) ALOX5GNRHRNAMPTTP53MAPT
SCHEMBL7081725 0.90 TP53 (0.32) ALOX5TP53POLBTHRBTLR7
SCHEMBL7085972 0.89 GRIN1 (0.37) GNRHRNAMPTPOLBTHRBTLR7
SCHEMBL6964165 0.87 POLB (0.38) ALOX5GNRHRTP53MAPTPOLB
SCHEMBL6966552 0.87 ENPP2 (0.31) GNRHRENPP2
SCHEMBL7082084 0.86 ENPP2 (0.35) NAMPTTP53MAPTPOLBENPP2
SCHEMBL6972096 0.85 LMNA (0.37) NAMPTTP53POLBTHRB
SCHEMBL6968974 0.85 ALDH1A1 (0.31) MAPT
SCHEMBL6974781 0.85 ENPP2 (0.35) NAMPTTP53MAPTPOLBTHRB
SCHEMBL7080069 0.84 S1PR3 (0.37) GNRHRTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed