SCHEMBL6973129

SCHEMBL6973129

CC(=O)OCCOCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MDM2 Q00987 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HDAC1 Q13547 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
S1PR3 Q99500 1/20 0.34
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CHRNA7 P36544 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRA5 P31644 1/20 0.33
CYP3A4 P08684 1/20 0.33
NOX4 Q9NPH5 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960297 0.92 MDM2 (0.34) ALDH1A1KDM4EMDM2KMT2AHDAC1
SCHEMBL7084562 0.92 KDM4E (0.37) ALDH1A1KDM4EMDM2KMT2AMEN1
SCHEMBL6969306 0.92 KMT2A (0.39) ALDH1A1KDM4EMDM2KMT2AMEN1
SCHEMBL6975778 0.90 MEN1 (0.36) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL6960775 0.90 GRIN1 (0.35) ALDH1A1KMT2AS1PR3
SCHEMBL7084645 0.90 ALDH1A1 (0.38) ALDH1A1KMT2AGABRA1GABRA5
SCHEMBL6969211 0.90 KMT2A (0.34) ALDH1A1KMT2AMEN1S1PR3GABRA1
SCHEMBL7082204 0.90 GRIN1 (0.35) S1PR3NOX4
SCHEMBL7085466 0.88 ALOX5AP (0.34) ALDH1A1KDM4EMDM2KMT2AHDAC1
SCHEMBL6962569 0.88 RXFP1 (0.38) ALDH1A1KDM4ECYP2C9CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed