SCHEMBL6975778

SCHEMBL6975778

CC(=O)OCCOCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
GSK3B P49841 1/20 0.33
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
AGTR1 P30556 1/20 0.31
AGTR2 P50052 1/20 0.31
ENPP2 Q13822 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HIF1A Q16665 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
PIM1 P11309 1/20 0.31
PIM3 Q86V86 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084824 0.92 PIM1 (0.34) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL6975053 0.92 MEN1 (0.41) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL6973001 0.91 P2RX3 (0.33) KMT2AGSK3BTP53
SCHEMBL6973129 0.90 ALDH1A1 (0.35) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL7086007 0.90 GRIN1 (0.33) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL6973843 0.89 TLR8 (0.32) MEN1KMT2A
SCHEMBL6973130 0.89 ENPP2 (0.32) MEN1KMT2AENPP2
SCHEMBL6967059 0.88 MAPT (0.33) CYP1A2CYP2C9CYP2C19GSK3BCYP3A4
SCHEMBL6967391 0.88 KMT2A (0.35) MEN1KMT2ACYP2C9CYP2C19CYP2D6
SCHEMBL7086333 0.87 CYP1A2 (0.39) MEN1KMT2ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed