SCHEMBL7084645

SCHEMBL7084645

CC(=O)OCCOCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
MCL1 Q07820 4/20 0.34
TP53 P04637 1/20 0.34
NPC1 O15118 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
PKM P14618 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
KMT2A Q03164 1/20 0.33
GRM5 P41594 1/20 0.33
GABRA5 P31644 3/20 0.32
GABRA1 P14867 2/20 0.32
SLC16A3 O15427 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969211 0.94 KMT2A (0.34) ALDH1A1MCL1TP53PKMOPRM1
SCHEMBL6969475 0.93 ALDH1A1 (0.37) ALDH1A1LMNAMCL1TP53NPC1
SCHEMBL7086211 0.93 ALDH1A1 (0.39) ALDH1A1LMNAMCL1TP53NPC1
SCHEMBL6967425 0.93 ALDH1A1 (0.40) ALDH1A1LMNATP53NPC1GRIN1
SCHEMBL6973001 0.92 P2RX3 (0.33) LMNATP53KMT2A
SCHEMBL6960775 0.91 GRIN1 (0.35) ALDH1A1LMNAGRIN1GRIN2BKMT2A
SCHEMBL6973129 0.90 ALDH1A1 (0.35) ALDH1A1KMT2AGABRA5GABRA1
SCHEMBL6972360 0.90 ALDH1A1 (0.37) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL6962569 0.89 RXFP1 (0.38) ALDH1A1LMNA
SCHEMBL7082204 0.87 GRIN1 (0.35) GRIN1GRIN2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed