SCHEMBL6969306

SCHEMBL6969306

CC(=O)OCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
S1PR3 Q99500 1/20 0.36
CYP3A4 P08684 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRA5 P31644 1/20 0.35
LMNA P02545 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MDM2 Q00987 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973129 0.92 ALDH1A1 (0.35) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL7086385 0.92 TLR7 (0.35) KMT2AALDH1A1KDM4EL3MBTL1S1PR3
SCHEMBL7084562 0.91 KDM4E (0.37) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL6964229 0.90 TOP2A (0.41) L3MBTL1S1PR3CYP3A4
SCHEMBL6967425 0.89 ALDH1A1 (0.40) KMT2AALDH1A1S1PR3GABRA1GABRA5
SCHEMBL6972338 0.89 GRIN1 (0.38) KMT2AALDH1A1S1PR3LMNAPKM
SCHEMBL6975053 0.89 MEN1 (0.41) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL6973275 0.89 ALDH1A1 (0.36) KMT2AMEN1ALDH1A1S1PR3GABRA1
SCHEMBL7079752 0.89 GRIN1 (0.37) ALDH1A1KDM4ES1PR3PKMSMN1; SMN2
SCHEMBL6972994 0.87 RXFP1 (0.41) KMT2AALDH1A1KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed