SCHEMBL6973165

SCHEMBL6973165

CC(C)c1nc(CN=C(N)N)n(Cc2ccccn2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 9/20 0.34
OPRM1 P35372 1/20 0.32
RIPK3 Q9Y572 1/20 0.32
GRIN1 Q05586 3/20 0.32
GRIN2B Q13224 3/20 0.32
TLR7 Q9NYK1 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GFER P55789 1/20 0.31
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30
PLA2G2A P14555 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078156 0.93 GRIN1 (0.36) S1PR3OPRM1RIPK3GRIN1GRIN2B
SCHEMBL6973295 0.89 HRH4 (0.34) GRIN1GRIN2BTLR7HRH4ALDH1A1
SCHEMBL6967022 0.89 ADRA1D (0.34) S1PR3GRIN1GRIN2BTLR7HRH4
SCHEMBL7078209 0.88 S1PR3 (0.34) S1PR3GRIN1GRIN2BTLR7KDM4E
SCHEMBL6973511 0.88 S1PR3 (0.36) S1PR3GRIN1GRIN2BTLR7KDM4E
SCHEMBL6969106 0.86 HRH1 (0.36) S1PR3OPRM1GRIN1GRIN2BTLR7
SCHEMBL6967358 0.86 S1PR3 (0.35) S1PR3GRIN1GRIN2BTLR7KDM4E
SCHEMBL6970221 0.85 S1PR3 (0.41) S1PR3ALDH1A1
SCHEMBL6957969 0.85 HTR3E (0.35) GRIN1GRIN2BHRH4KDM4EALDH1A1
SCHEMBL7084640 0.85 S1PR3 (0.39) S1PR3OPRM1TLR7KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed