SCHEMBL6973437

SCHEMBL6973437

CC(=O)NCc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.38
S1PR3 Q99500 7/20 0.37
NPC1 O15118 1/20 0.37
RHEB Q15382 1/20 0.36
HPGD P15428 1/20 0.35
TP53 P04637 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NTRK1 P04629 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969739 0.93 POLB (0.38) KMT2AALDH1A1S1PR3NPC1HPGD
SCHEMBL6962934 0.92 MEN1 (0.39) MEN1KMT2AALDH1A1S1PR3NPC1
SCHEMBL6965884 0.90 ALDH1A1 (0.41) KMT2AALDH1A1S1PR3NPC1TP53
SCHEMBL6973222 0.89 S1PR3 (0.41) ALDH1A1S1PR3NTRK1
SCHEMBL6974447 0.89 MEN1 (0.34) MEN1KMT2AALDH1A1S1PR3RHEB
SCHEMBL6976953 0.87 ALDH1A1 (0.33) MEN1KMT2AALDH1A1S1PR3TP53
SCHEMBL7078972 0.86 SLC16A3 (0.35) MEN1KMT2AALDH1A1S1PR3NPC1
SCHEMBL6973271 0.86 POLB (0.35) MEN1KMT2AALDH1A1HPGDTP53
SCHEMBL7084143 0.86 S1PR3 (0.41) KMT2AALDH1A1S1PR3HPGDNTRK1
SCHEMBL8343030 0.85 LMNA (0.40) MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed