SCHEMBL6962934

SCHEMBL6962934

CC(C)c1nc(CNC(N)=O)n(Cc2ccccn2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.37
ADRA1D P25100 1/20 0.37
S1PR3 Q99500 7/20 0.36
NPC1 O15118 1/20 0.36
RHEB Q15382 1/20 0.36
XIAP P98170 1/20 0.35
BIRC2 Q13490 1/20 0.35
BACE1 P56817 1/20 0.35
HPGD P15428 1/20 0.35
TP53 P04637 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085418 0.93 POLB (0.38) KMT2AALDH1A1ADRA1DS1PR3NPC1
SCHEMBL6973437 0.92 MEN1 (0.40) MEN1KMT2AALDH1A1S1PR3NPC1
SCHEMBL7082911 0.90 ALDH1A1 (0.40) MEN1KMT2AALDH1A1S1PR3NPC1
SCHEMBL6970221 0.89 S1PR3 (0.41) ALDH1A1S1PR3
SCHEMBL6974447 0.88 MEN1 (0.34) MEN1KMT2AALDH1A1S1PR3RHEB
SCHEMBL6966022 0.87 ADRA1D (0.36) MEN1KMT2AALDH1A1ADRA1DS1PR3
SCHEMBL6970129 0.86 S1PR3 (0.40) KMT2AALDH1A1S1PR3HPGD
SCHEMBL6975001 0.86 ALDH1A1 (0.33) MEN1KMT2AALDH1A1ADRA1DXIAP
SCHEMBL6976953 0.86 ALDH1A1 (0.33) MEN1KMT2AALDH1A1ADRA1DS1PR3
SCHEMBL6973271 0.86 POLB (0.35) MEN1KMT2AALDH1A1HPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed