SCHEMBL6974966

SCHEMBL6974966

CC(C)c1nc(CCOC(N)=O)n(Cc2cccnc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
IDO1 P14902 1/20 0.34
S1PR3 Q99500 4/20 0.34
GRM2 Q14416 2/20 0.34
ENPP2 Q13822 1/20 0.33
TLR7 Q9NYK1 4/20 0.33
PKM P14618 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970826 0.95 GRIN1 (0.35) GRIN1GRIN2BIDO1S1PR3GRM2
SCHEMBL7080841 0.94 GRIN1 (0.36) GRIN1GRIN2BIDO1S1PR3GRM2
SCHEMBL6973065 0.93 GRIN1 (0.35) GRIN1GRIN2BIDO1S1PR3GRM2
SCHEMBL6972580 0.92 GRIN1 (0.36) GRIN1GRIN2BIDO1S1PR3ENPP2
SCHEMBL6967126 0.92 GRIN1 (0.37) GRIN1GRIN2BIDO1S1PR3GRM2
SCHEMBL6973955 0.91 ALDH1A1 (0.35) S1PR3TLR7HDAC1HDAC8
SCHEMBL6967887 0.91 LMNA (0.35) ENPP2TLR7
SCHEMBL6966178 0.90 ADRA1D (0.36) S1PR3
SCHEMBL6967988 0.90 ENPP2 (0.35) ENPP2
SCHEMBL6974469 0.90 TLR7 (0.36) S1PR3ENPP2TLR7HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed