SCHEMBL6973574

SCHEMBL6973574

CC(C)c1c(Sc2cccc(Cl)c2)nc(CN)n1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
MEN1 O00255 3/20 0.41
KDM4E B2RXH2 2/20 0.41
PTPN11 Q06124 2/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAOB P27338 2/20 0.38
MAOA P21397 1/20 0.38
MAPT P10636 3/20 0.37
GRM5 P41594 3/20 0.36
EGFR P00533 1/20 0.36
LCK P06239 1/20 0.36
POLB P06746 1/20 0.35
DHFR P00374 1/20 0.35
PPP1CA P62136 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972112 0.88 LMNA (0.39) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL6974384 0.87 HSP90B1 (0.34) PTPN11
SCHEMBL6961944 0.86 ALDH1A1 (0.40) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL7080119 0.85 MAOA (0.38) ALDH1A1MAOBMAOA
SCHEMBL6961421 0.84 SLC6A4 (0.36) KMT2AALDH1A1KDM4EPTPN11LMNA
SCHEMBL6969756 0.82 ALOX12 (0.40) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL6970165 0.82 ALDH1A1 (0.43) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL6964412 0.81 ALOX12 (0.41) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL6973812 0.81 LMNA (0.39) KMT2AALDH1A1HPGDMEN1KDM4E
SCHEMBL6964721 0.81 ALDH1A1 (0.35) KMT2AALDH1A1HPGDMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed