SCHEMBL6973592

SCHEMBL6973592

Nc1ccc(Sc2cccc3cnccc23)c([N+](=O)[O-])c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HASPIN Q8TF76 6/20 0.42
GSK3B P49841 1/20 0.42
CLK1 P49759 1/20 0.41
MAPT P10636 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PSMD14 O00487 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963335 0.80 LMNA (0.46) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6968103 0.80 MAPT (0.48) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6972315 0.80 LMNA (0.46) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6973656 0.76 PDE7A (0.60) LMNAMAPTMEN1KMT2ANPSR1
SCHEMBL6963693 0.76 MAPT (0.60) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6958268 0.76 LMNA (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6965142 0.76 PDE7A (0.47) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6958271 0.76 LMNA (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6965245 0.76 LMNA (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6968741 0.76 KDM4E (0.57) LMNACYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed