SCHEMBL6965787

SCHEMBL6965787

CC(C)c1nc(CN)n(Cc2cccnc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
LMNA P02545 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
P2RX7 Q99572 2/20 0.37
GABRA5 P31644 3/20 0.36
KDM4E B2RXH2 3/20 0.36
HTT P42858 2/20 0.36
TSHR P16473 2/20 0.36
GABRA1 P14867 2/20 0.36
TP53 P04637 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
KMT2A Q03164 2/20 0.35
PKM P14618 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971118 0.93 ALDH1A1 (0.37) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6957238 0.92 GABRA5 (0.36) ALDH1A1GRIN1GRIN2BP2RX7GABRA5
SCHEMBL6970034 0.90 ALDH1A1 (0.40) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6967360 0.90 IDO1 (0.36) ALDH1A1KDM4EHTTSMN1; SMN2TDP1
SCHEMBL6962312 0.89 HTR3E (0.40) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL7085996 0.89 ALDH1A1 (0.39) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6974922 0.89 POLB (0.41) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6965333 0.89 ALDH1A1 (0.41) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6974887 0.89 GRIN1 (0.39) ALDH1A1GRIN1GRIN2BKDM4EHPGD
SCHEMBL6972848 0.88 TLR7 (0.38) ALDH1A1P2RX7GABRA5KDM4EGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed