SCHEMBL6970034

SCHEMBL6970034

CC(C)c1nc(CO)n(Cc2cccnc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
LMNA P02545 2/20 0.40
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
P2RX7 Q99572 1/20 0.37
GABRA5 P31644 2/20 0.36
KDM4E B2RXH2 2/20 0.36
HTT P42858 2/20 0.36
TP53 P04637 2/20 0.36
TSHR P16473 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GABRA1 P14867 1/20 0.36
SRC P12931 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
PKM P14618 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085996 0.93 ALDH1A1 (0.39) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6973652 0.92 SRC (0.37) ALDH1A1GRIN1GRIN2BGABRA5KDM4E
SCHEMBL7084751 0.91 ALDH1A1 (0.38) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6965787 0.90 ALDH1A1 (0.38) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL7079909 0.90 IDO1 (0.36) ALDH1A1KDM4ETP53SMN1; SMN2TDP1
SCHEMBL6975192 0.90 TDP1 (0.43) ALDH1A1LMNAKDM4ETP53TDP1
SCHEMBL6962312 0.89 HTR3E (0.40) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6965333 0.89 ALDH1A1 (0.41) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6971118 0.89 ALDH1A1 (0.37) ALDH1A1LMNAGRIN1GRIN2BP2RX7
SCHEMBL6974922 0.89 POLB (0.41) ALDH1A1LMNAGRIN1GRIN2BP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed