SCHEMBL6973420

SCHEMBL6973420

CC(=O)OCCOC(Cc1ccccn1)c1nc(C(C)C)c(Sc2cccc(Cl)c2)[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SLC6A9 P48067 4/20 0.34
ALDH1A1 P00352 1/20 0.32
PPP1CA P62136 1/20 0.32
KMT2A Q03164 1/20 0.32
GRM5 P41594 1/20 0.32
TP53 P04637 2/20 0.31
RXFP1 Q9HBX9 1/20 0.31
CACNA1B Q00975 1/20 0.31
PGR P06401 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
PTGS1 P23219 1/20 0.31
SLC6A2 P23975 1/20 0.31
MDM2 Q00987 1/20 0.31
POLB P06746 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087680 0.94 MEN1 (0.33) SMN1; SMN2NPC1KMT2APGRADORA3
SCHEMBL7080029 0.91 PTPRA (0.34) SMN1; SMN2MAPTNPC1ALDH1A1PGR
SCHEMBL7078551 0.91 SLC6A9 (0.33) SLC6A9KMT2APGRADORA3PTGS1
SCHEMBL6960274 0.89 MAPT (0.34) SMN1; SMN2MAPTNPC1RAB9ASLC6A9
SCHEMBL7081154 0.89 MAPT (0.35) SMN1; SMN2MAPTNPC1RAB9ASLC6A9
SCHEMBL6975428 0.88 CYP1A2 (0.35) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL8113590 0.87 MAOB (0.32) PGRADORA3PTGS1SLC6A2
SCHEMBL6973004 0.87 SLC6A9 (0.32) SLC6A9KMT2ATP53RXFP1
SCHEMBL7086458 0.87 TP53 (0.36) SLC6A9TP53RXFP1
SCHEMBL7084647 0.85 ALDH1A1 (0.38) SMN1; SMN2NPC1RAB9ASLC6A9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed