SCHEMBL7080029

SCHEMBL7080029

CC(=O)OCCOC(Cc1ccccn1)c1nc(C(C)C)c(Sc2ccccc2)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.34
PGR P06401 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A2 P23975 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
CYP1A2 P05177 3/20 0.31
TSHR P16473 2/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HTT P42858 1/20 0.31
ATM Q13315 1/20 0.31
NPC1 O15118 1/20 0.31
HDAC6 Q9UBN7 4/20 0.30
HDAC1 Q13547 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078551 0.91 SLC6A9 (0.33) PGRADORA3PTGS1SLC6A2
SCHEMBL6973420 0.91 SMN1; SMN2 (0.35) PTPRAPGRADORA3PTGS1SLC6A2
SCHEMBL7087680 0.91 MEN1 (0.33) PGRADORA3PTGS1SLC6A2TAS1R3
SCHEMBL8113590 0.91 MAOB (0.32) PGRADORA3PTGS1SLC6A2HDAC6
SCHEMBL6975428 0.88 CYP1A2 (0.35) CYP1A2TSHRCYP2D6MAPTSMN1; SMN2
SCHEMBL7084495 0.88 PTPRA (0.37) PTPRAPGRADORA3PTGS1SLC6A2
SCHEMBL6974559 0.88 PTPRA (0.32) PTPRA
SCHEMBL6975782 0.86 CDK5 (0.33) CYP1A2CYP2D6ALDH1A1
SCHEMBL7086334 0.86 DHFR (0.32) CYP1A2ALDH1A1
SCHEMBL6973132 0.84 LMNA (0.34) CYP1A2SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed