SCHEMBL6975998

SCHEMBL6975998

CC1=C(C)C2=C(N)C(C)(CN3CCN(C(=O)C(c4ccccc4)c4ccccc4)CC3)CC2=C(C)O1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 4/20 0.41
LMNA P02545 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HTT P42858 2/20 0.39
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
GAA P10253 2/20 0.37
TP53 P04637 1/20 0.37
P2RX7 Q99572 1/20 0.36
CYP2D6 P10635 1/20 0.36
ADRB2 P07550 1/20 0.36
CHRM1 P11229 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980783 0.88 CACNA2D1 (0.43)
SCHEMBL6983252 0.87 CACNA1B (0.36) OPRK1
Hydrochloric Acid SCHEMBL6984864 0.82 OPRL1 (0.38) CYP2D6OPRK1
SCHEMBL6977659 0.82 L3MBTL1 (0.45) TSHRALDH1A1KDM4ELMNAMEN1
SCHEMBL6981795 0.80 POLB (0.47) TSHRALDH1A1KDM4ELMNAMEN1
SCHEMBL6974103 0.80 NPC1 (0.48) TSHRALDH1A1KDM4ENPSR1HTT
SCHEMBL6984706 0.79 ALDH1A1 (0.40) ALDH1A1KDM4ELMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL6984801 0.79 SMN1; SMN2 (0.43) TSHRALDH1A1LMNANPSR1MEN1
SCHEMBL6976601 0.77 KCNA3 (0.41)
SCHEMBL6983932 0.77 CHRM2 (0.43) LMNAHTTCYP2D6CHRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed