SCHEMBL6980783

SCHEMBL6980783

CC1=C(C)C2=C(N)C(C)(CN3CCN(C(=O)CC(c4ccccc4)c4ccccc4)CC3)CC2=C(C)O1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 12/20 0.43
CACNA1B Q00975 12/20 0.43
CACNB1 Q02641 12/20 0.43
CACNA1C Q13936 10/20 0.43
CACNA1H O95180 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
CACNA1G O43497 5/20 0.40
KCNH2 Q12809 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983252 0.92 CACNA1B (0.36) CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL6975998 0.88 TSHR (0.44)
SCHEMBL6977659 0.85 L3MBTL1 (0.45) TDP1
SCHEMBL6974103 0.83 NPC1 (0.48) CACNA1CTDP1
Hydrochloric Acid SCHEMBL6984864 0.83 OPRL1 (0.38)
Hydrochloric Acid SCHEMBL6982807 0.82 SIGMAR1 (0.42) KCNH2
SCHEMBL6984706 0.79 ALDH1A1 (0.40)
Hydrochloric Acid SCHEMBL6984801 0.78 SMN1; SMN2 (0.43) KCNH2
SCHEMBL6981795 0.78 POLB (0.47)
SCHEMBL6981070 0.77 SIGMAR1 (0.41) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed