SCHEMBL6977058

SCHEMBL6977058

CC1CCN(C(=O)CCc2ccc(C#N)cc2)c2c(N)cccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.36
KDM1A O60341 5/20 0.36
YAP1 P46937 1/20 0.36
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PRKAA2 P54646 1/20 0.35
KCNJ1 P48048 1/20 0.34
KCNH2 Q12809 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTR1A P08908 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
OPRM1 P35372 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985050 0.80 ALDH1A1 (0.39) YAP1ALDH1A1MEN1TSHRKMT2A
SCHEMBL6977052 0.80 TP53 (0.39) KDM1AYAP1SMN1; SMN2KCNJ1KCNH2
SCHEMBL6974890 0.78 DPP8 (0.37) FFAR1KDM1AYAP1HPGDSMN1; SMN2
SCHEMBL6979727 0.78 TSHR (0.40) FFAR1HPGDSMN1; SMN2KCNJ1KCNH2
SCHEMBL6980061 0.73 KCNJ1 (0.47) FFAR1HPGDSMN1; SMN2KCNJ1KCNH2
SCHEMBL6985046 0.70 KMT2A (0.43) SMN1; SMN2ALDH1A1MAPK1HTR2AMEN1
SCHEMBL6974883 0.69 TP53 (0.41) FFAR1KDM1ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL7410532 0.69 CHRM2 (0.41) KDM1AYAP1HPGDSMN1; SMN2ALDH1A1
SCHEMBL6986713 0.68 TSHR (0.41) FFAR1HPGDKCNJ1KCNH2ALDH1A1
SCHEMBL6986437 0.67 PTGER4 (0.41) FFAR1HPGDSMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed