SCHEMBL6986437

SCHEMBL6986437

CNc1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
ATM Q13315 1/20 0.39
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
FPR1 P21462 2/20 0.39
FPR2 P25090 2/20 0.39
TSHR P16473 3/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980994 0.86 RXRA (0.43) PTGER4HDAC6ATMMAPTNPC1
SCHEMBL6978509 0.86 PTGER4 (0.40) PTGER4HDAC1HDAC8HDAC6ATM
SCHEMBL6977736 0.86 CHRM3 (0.40) PTGER4ATMMAPTNPC1MAPK1
SCHEMBL6984462 0.85 ATM (0.41) PTGER4HDAC1HDAC8HDAC6ATM
SCHEMBL6985381 0.85 MMP1 (0.45) PTGER4HDAC1HDAC8HDAC6ATM
SCHEMBL6982945 0.85 NR3C1 (0.36) PTGER4ATMMAPTNPC1MAPK1
SCHEMBL6986817 0.85 THRB (0.42) HDAC1HDAC8HDAC6ATMMAPT
SCHEMBL6976287 0.84 NOTUM (0.38) PTGER4HDAC1HDAC8HDAC6ATM
SCHEMBL6979727 0.84 TSHR (0.40) PTGER4HDAC1HDAC8HDAC6MAPT
SCHEMBL6985248 0.84 MAPT (0.42) PTGER4MAPTNPC1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed