SCHEMBL6978201

SCHEMBL6978201

O=C(CC(=O)C(F)F)c1nc2ccccc2s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.60
NPC1 O15118 5/20 0.60
SMN1; SMN2 Q16637 4/20 0.60
HPGD P15428 3/20 0.60
ALDH1A1 P00352 4/20 0.55
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
CASP1 P29466 1/20 0.55
PKM P14618 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
MAPT P10636 3/20 0.52
LMNA P02545 2/20 0.51
TP53 P04637 1/20 0.51
GAA P10253 1/20 0.51
MCL1 Q07820 1/20 0.51
HTR1A P08908 2/20 0.48
DRD2 P14416 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7584707 0.84 NPC1 (0.56) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL23617613 0.81 NPC1 (0.63) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6979336 0.81 PDPK1 (0.50) SMN1; SMN2HPGDALDH1A1PKMMAPT
SCHEMBL6979211 0.81 RAB9A (0.58) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6984031 0.80 ACP1 (0.50) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6983145 0.80 DYRK1A (0.49) RAB9ANPC1SMN1; SMN2ALDH1A1NFKB1
SCHEMBL6972342 0.80 RAB9A (0.39) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6975021 0.79 ALOX5 (0.44) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6971921 0.79 LMNA (0.39) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL6978735 0.78 GAA (0.48) RAB9ANPC1SMN1; SMN2HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed