SCHEMBL6972342

SCHEMBL6972342

O=C(CC(=O)C(F)F)c1nc2cccc(F)c2s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.39
NPC1 O15118 5/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HPGD P15428 1/20 0.39
MAOB P27338 3/20 0.37
AKR1A1 P14550 1/20 0.37
AKR1B1 P15121 1/20 0.37
NAAA Q02083 1/20 0.37
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
MCL1 Q07820 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971921 0.85 LMNA (0.39) RAB9ANPC1SMN1; SMN2HPGDMAOB
SCHEMBL6975021 0.85 ALOX5 (0.44) RAB9ANPC1SMN1; SMN2HPGDMAOB
SCHEMBL6972014 0.81 PLOD2 (0.41) RAB9ANPC1SMN1; SMN2HPGDMAOB
SCHEMBL6978201 0.80 RAB9A (0.60) RAB9ANPC1SMN1; SMN2HPGDMAOB
SCHEMBL6978735 0.80 GAA (0.48) RAB9ANPC1SMN1; SMN2HPGDMAPT
SCHEMBL7960065 0.76 AKR1A1 (0.43) RAB9ANPC1SMN1; SMN2HPGDMAOB
SCHEMBL19691127 0.75 DYRK1A (0.43) RAB9ANPC1SMN1; SMN2MAOBAKR1A1
SCHEMBL6977213 0.75 GAA (0.40) RAB9ANPC1SMN1; SMN2AKR1A1AKR1B1
SCHEMBL6979336 0.74 PDPK1 (0.50) SMN1; SMN2HPGDMAOBMAPTALDH1A1
SCHEMBL6983145 0.70 DYRK1A (0.49) RAB9ANPC1SMN1; SMN2MAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed