SCHEMBL6978353

SCHEMBL6978353

CCCCCCCN1CCC(C[C@H](O)Cc2ccnc3c(OC)cccc23)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 3/20 0.46
HTR4 Q13639 3/20 0.45
HTR1D P28221 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
HTR2B P41595 1/20 0.45
HTR1A P08908 2/20 0.41
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
CHRM5 P08912 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KCNH2 Q12809 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977618 0.85 HTR4 (0.46) ADRB3HTR4HTR1DHTR2AHTR7
SCHEMBL6975733 0.83 HTR4 (0.48) HTR4HTR1DHTR2AHTR7HTR2B
SCHEMBL6977170 0.80 CCR8 (0.53) CHRM2KDM4EALDH1A1KCNH2MEN1
SCHEMBL6977177 0.80 CCR8 (0.53) CHRM2KDM4EALDH1A1KCNH2MEN1
SCHEMBL6977174 0.80 CCR8 (0.53) CHRM2KDM4EALDH1A1KCNH2MEN1
SCHEMBL6976945 0.80 HTR4 (0.57) HTR4HTR1DHTR2AHTR7HTR2B
SCHEMBL6628061 0.80 HTR1A (0.54) HTR4HTR1DHTR2AHTR7HTR2B
SCHEMBL6973562 0.76 HTR4 (0.46) ADRB3HTR4HTR1DHTR2AHTR7
SCHEMBL6626086 0.76 HTR1A (0.47) HTR4HTR1DHTR2AHTR7HTR2B
SCHEMBL6970302 0.74 ADRA1A (0.48) HTR1ACHRM3KDM4EALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP claimed