SCHEMBL6978428

SCHEMBL6978428

Cc1c(C)c2c(c(C)c1NC(=O)O)CC(C)(CCN1CCC(OC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 10/20 0.44
CHRM2 P08172 2/20 0.43
HTR1A P08908 2/20 0.43
ADRA2A P08913 2/20 0.43
CHRM1 P11229 2/20 0.43
DRD1 P21728 2/20 0.43
SLC6A2 P23975 2/20 0.43
ADRA1A P35348 2/20 0.43
DRD3 P35462 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 2/20 0.43
NPC1 O15118 1/20 0.43
MLNR O43193 1/20 0.43
NR1I2 O75469 1/20 0.43
EGFR P00533 1/20 0.43
LMNA P02545 1/20 0.43
ERBB2 P04626 1/20 0.43
FYN P06241 1/20 0.43
CHRM4 P08173 1/20 0.43
ABCB1 P08183 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985715 0.88 KCNA3 (0.42) SLC6A2SLC6A3SLC6A4
Oxalic Acid SCHEMBL6983672 0.87 BCHE (0.43) BCHECHRM2HTR1AADRA2ACHRM1
SCHEMBL6985682 0.87 SLC6A4 (0.49) SLC6A2SLC6A3SLC6A4
SCHEMBL6979549 0.86 CHRM2 (0.44) BCHECHRM2HTR1AADRA2ACHRM1
Oxalic Acid SCHEMBL6980644 0.78 GRM5 (0.42) BCHECHRM2HTR1AADRA2ACHRM1
SCHEMBL6983930 0.77 CHRM2 (0.43) BCHECHRM2HTR1AADRA2ACHRM1
Oxalic Acid SCHEMBL6984301 0.74 SLC6A4 (0.53) SLC6A2SLC6A3SLC6A4
SCHEMBL6982775 0.74 SLC6A3 (0.37) BCHESLC6A2SLC6A3LMNASLC6A4
SCHEMBL6984905 0.74 KCNA3 (0.44) SLC6A2SLC6A3SLC6A4
SCHEMBL6980736 0.73 ACHE (0.38) BCHEKCNH2ACHEEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed