SCHEMBL6980093

SCHEMBL6980093

C[S+]([O-])c1ccc(-c2oc3cc(F)ccc3c(=O)c2-c2ccccc2F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.43
MAPK14 Q16539 3/20 0.42
NMUR2 Q9GZQ4 1/20 0.41
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
MAOB P27338 2/20 0.38
NTRK1 P04629 1/20 0.38
PLK3 Q9H4B4 1/20 0.38
PLA2G2A P14555 1/20 0.37
PLA2G4A P47712 1/20 0.37
PTGS1 P23219 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983326 0.87 MAPK14 (0.49) PTGS2MAPK14ACHEBACE1MAOB
SCHEMBL6982162 0.85 PTGS2 (0.44) PTGS2MAPK14ACHEBACE1MAOB
SCHEMBL6981848 0.81 MAPK14 (0.40) PTGS2MAPK14ACHEBACE1MAOB
SCHEMBL6972864 0.81 PTGS2 (0.59) PTGS2MAPK14NMUR2NTRK1PLK3
SCHEMBL6972243 0.74 PTGS2 (0.68) PTGS2MAPK14NMUR2NTRK1PLK3
SCHEMBL6977374 0.73 GABRP (0.41) PTGS2MAPK14ACHEBACE1CYP3A4
SCHEMBL6978136 0.71 PTGS2 (0.68) PTGS2MAPK14NMUR2NTRK1PLK3
SCHEMBL6974299 0.71 PTGS2 (0.67) PTGS2MAPK14NTRK1PLK3PTGS1
SCHEMBL6976415 0.69 PTGS2 (0.67) PTGS2MAPK14NMUR2NTRK1PLK3
SCHEMBL6979230 0.67 PTGS2 (0.65) PTGS2MAPK14MAOBPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105384-B1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-03-26 EP disclosed
US-6340694-B1 Diarylbenzopyran derivatives as cyclooxygenase-2 inhibitors PACIFIC CORPORATION (KR) 2002-01-22 US disclosed
EP-1105384-A1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-13 EP disclosed
WO-2000010993-A1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-03-02 WO disclosed