SCHEMBL6981848

SCHEMBL6981848

C[S+]([O-])c1ccc(-c2oc3cc(F)ccc3c(=O)c2-c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.40
PTGS2 P35354 6/20 0.39
PTGS1 P23219 2/20 0.39
MAOB P27338 2/20 0.36
ACHE P22303 2/20 0.36
BACE1 P56817 2/20 0.36
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
PLA2G2A P14555 1/20 0.34
PLA2G4A P47712 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983326 0.89 MAPK14 (0.49) MAPK14PTGS2PTGS1MAOBACHE
SCHEMBL6982162 0.87 PTGS2 (0.44) MAPK14PTGS2PTGS1MAOBACHE
SCHEMBL6981239 0.81 PTGS1 (0.52) MAPK14PTGS2PTGS1MAOBCA1
SCHEMBL6980093 0.81 PTGS2 (0.43) MAPK14PTGS2PTGS1MAOBACHE
SCHEMBL6977374 0.72 GABRP (0.41) MAPK14PTGS2ACHEBACE1KDM4E
SCHEMBL6972219 0.70 PTGS2 (0.66) MAPK14PTGS2PTGS1PLA2G2APLA2G4A
SCHEMBL6973900 0.69 PTGS2 (0.50) MAPK14PTGS2PTGS1
SCHEMBL6979230 0.69 PTGS2 (0.65) MAPK14PTGS2PTGS1MAOB
SCHEMBL6982972 0.68 PTGS2 (0.57) MAPK14PTGS2PTGS1MAOBCA2
SCHEMBL6971292 0.68 PTGS2 (0.65) MAPK14PTGS2PTGS1MAOBCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105384-B1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-03-26 EP disclosed
US-6340694-B1 Diarylbenzopyran derivatives as cyclooxygenase-2 inhibitors PACIFIC CORPORATION (KR) 2002-01-22 US disclosed
EP-1105384-A1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-13 EP disclosed
WO-2000010993-A1 DIARYLBENZOPYRAN DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-03-02 WO disclosed