SCHEMBL6980127

SCHEMBL6980127

N#Cc1ccc(CCC(=O)N2CCCc3cc(N(CCc4ccccc4)S(=O)(=O)c4ccccc4)ccc32)cc1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 8/20 0.53
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
TP53 P04637 1/20 0.42
LMNA P02545 1/20 0.42
KDM1A O60341 2/20 0.41
POLB P06746 1/20 0.41
NR1I2 O75469 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977634 0.88 NR3C1 (0.53) NR3C1ALDH1A1MEN1HPGDKMT2A
SCHEMBL6987763 0.87 NR3C1 (0.47) NR3C1ALDH1A1GAAHPGDLMNA
Hydrochloric Acid SCHEMBL6984704 0.86 NR3C1 (0.49) NR3C1ALDH1A1GAAMEN1HPGD
SCHEMBL6987628 0.86 NR3C1 (0.48) NR3C1ALDH1A1MEN1HPGDKMT2A
SCHEMBL6982667 0.84 NR3C1 (0.41) NR3C1ALDH1A1GAAMEN1HPGD
SCHEMBL6983746 0.82 NR3C1 (0.47) NR3C1ALDH1A1GAAMEN1HPGD
SCHEMBL6985998 0.82 NR3C1 (0.47) NR3C1ALDH1A1GAAMEN1HPGD
SCHEMBL6986006 0.81 NR3C1 (0.46) NR3C1ALDH1A1GAAMEN1HPGD
SCHEMBL6979167 0.80 KDM1A (0.47) NR3C1ALDH1A1MEN1HPGDKMT2A
SCHEMBL7956609 0.79 NR3C1 (0.44) NR3C1ALDH1A1GAAMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed