SCHEMBL6982667

SCHEMBL6982667

N#Cc1ccc(CCC(=O)N2CCCc3cccc(N(CCc4ccccc4)S(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 4/20 0.41
TAS2R14 Q9NYV8 1/20 0.40
ALDH1A1 P00352 4/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
POLB P06746 1/20 0.38
AR P10275 1/20 0.37
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
TP53 P04637 2/20 0.35
PGR P06401 1/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
LMNA P02545 1/20 0.35
NR1I2 O75469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977636 0.90 ALDH1A1 (0.42) NR3C1TAS2R14ALDH1A1ARMEN1
SCHEMBL6987767 0.86 TP53 (0.42) NR3C1ALDH1A1KEAP1NFE2L2GAA
SCHEMBL6987632 0.85 ALDH1A1 (0.39) NR3C1TAS2R14ALDH1A1POLBMEN1
SCHEMBL6986002 0.84 RXRA (0.45) TAS2R14ALDH1A1ARMEN1HPGD
SCHEMBL6980127 0.84 NR3C1 (0.53) NR3C1ALDH1A1POLBMEN1HPGD
SCHEMBL6983751 0.82 NR3C1 (0.40) NR3C1ALDH1A1ARMEN1HPGD
SCHEMBL6986008 0.82 MEN1 (0.39) ALDH1A1MEN1HPGDKMT2AHSD17B10
SCHEMBL6979172 0.81 KDM1A (0.41) TAS2R14ALDH1A1MEN1HPGDKMT2A
SCHEMBL6981987 0.80 PTGER4 (0.38) NR3C1ALDH1A1ARMEN1HPGD
SCHEMBL6985322 0.80 GAA (0.41) NR3C1ALDH1A1ARMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed