SCHEMBL6981336

SCHEMBL6981336

CCCn1cc(-n2c(-c3cn(CCCCN4C(=O)c5ccccc5C4=O)c4ccccc34)c(C#N)n(C)c2=O)c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 3/20 0.42
CDK9 P50750 3/20 0.42
CCNA2 P20248 2/20 0.41
CDK2 P24941 2/20 0.41
CNR2 P34972 8/20 0.38
CNR1 P21554 2/20 0.37
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
MGAM O43451 2/20 0.36
GAA P10253 2/20 0.36
SI P14410 2/20 0.36
MGAM2 Q2M2H8 2/20 0.36
CAMK2D Q13557 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979460 0.89 CAMK2D (0.42) CCNT1CDK9CCNA2CDK2CNR2
SCHEMBL6978208 0.77 CNR1 (0.40) CCNT1CDK9CCNA2CDK2CNR2
SCHEMBL6980500 0.76 CCNT1 (0.41) CCNT1CDK9CCNA2CDK2CAMK2D
SCHEMBL6980479 0.74 CAMK2D (0.45) CCNT1CDK9CCNA2CDK2CAMK2D
SCHEMBL6985899 0.73 MAPT (0.40) CCNT1CDK9CCNA2CDK2CNR2
SCHEMBL6981135 0.71 ALDH1A1 (0.40) CCNT1CDK9CCNA2CDK2CNR1
Dimethylamine SCHEMBL6976140 0.69 CCNT1 (0.41) CCNT1CDK9CCNA2CDK2MGAM
Trifluoroacetic Acid SCHEMBL6985258 0.69 CAMK2D (0.39) CCNT1CDK9CCNA2CDK2CNR2
SCHEMBL7815250 0.66 MAPT (0.54) CNR2GLAMAPTMAPK1GAA
SCHEMBL6979590 0.66 CCNT1 (0.42) CCNT1CDK9CCNA2CDK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-B1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2003-08-27 EP disclosed
US-6346625-B1 ENZYME INHIBITORS FOR PROTEIN KINASES ASTRAZENECA AB (SE) 2002-02-12 US disclosed
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP disclosed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO disclosed