SCHEMBL6978208

SCHEMBL6978208

CCCn1cc(-n2c(-c3cn(CCCCN4C(=O)c5ccccc5C4=O)c4ccccc34)c(C(N)=O)[nH]c2=O)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.40
ICMT O60725 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CNR2 P34972 4/20 0.38
CCNT1 O60563 2/20 0.37
CDK9 P50750 2/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981421 0.87 ALDH1A1 (0.42) CNR1ALDH1A1MAPTNPSR1
SCHEMBL6981336 0.77 CCNT1 (0.42) CNR1ALDH1A1MAPTCNR2CCNT1
SCHEMBL6979608 0.76 CAMK2D (0.35) CNR1CA12CA1CA2CA9
SCHEMBL6985899 0.75 MAPT (0.40) CNR1ALDH1A1MAPTNPSR1CNR2
SCHEMBL6980479 0.75 CAMK2D (0.45) CCNT1CDK9CCNA2CDK2
SCHEMBL6981135 0.73 ALDH1A1 (0.40) CNR1CA12CA1CA2CA9
SCHEMBL7005339 0.73 CAMK2D (0.55)
SCHEMBL7005879 0.73 PIM1 (0.48) CNR1MAPTCCNT1CDK9CCNA2
Acetic Acid SCHEMBL7007558 0.72 CAMK2D (0.53)
Trifluoroacetic Acid SCHEMBL6985258 0.72 CAMK2D (0.39) CA12CA1CA2CA9CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-B1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2003-08-27 EP disclosed
US-6346625-B1 ENZYME INHIBITORS FOR PROTEIN KINASES ASTRAZENECA AB (SE) 2002-02-12 US disclosed