SCHEMBL6982164

SCHEMBL6982164

CC(OC(=O)CNc1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=N)N)cc1)S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.44
NR3C1 P04150 5/20 0.43
F2 P00734 6/20 0.40
PRSS1 P07477 4/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
MCL1 Q07820 1/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982167 0.83 F10 (0.44) F10NR3C1F2PRSS1PDE4A
Iodide SCHEMBL7956640 0.83 F10 (0.44) F10NR3C1F2PRSS1PDE4A
Hydrochloric Acid SCHEMBL6977280 0.82 NR3C1 (0.61) F10NR3C1F2PRSS1ALDH1A1
Hydrochloric Acid SCHEMBL7089726 0.81 FFAR1 (0.47) F10NR3C1F2PRSS1ALDH1A1
Hydrochloric Acid SCHEMBL6985379 0.79 ALDH1A1 (0.42) F10NR3C1F2PRSS1ALDH1A1
SCHEMBL6981023 0.78 RAB9A (0.45) F10NR3C1F2PRSS1ALDH1A1
Hydrochloric Acid SCHEMBL6981077 0.77 RAB9A (0.44) F10NR3C1F2PRSS1ALDH1A1
Hydrochloric Acid SCHEMBL6982225 0.77 PARP1 (0.39) F10NR3C1F2ALDH1A1GAA
SCHEMBL6982740 0.76 NR3C1 (0.59) NR3C1F2LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL6985423 0.76 NR3C1 (0.44) NR3C1ALDH1A1LMNAPKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed