SCHEMBL6983709

SCHEMBL6983709

N=C(N)c1ccc(NC(=O)CCC(=O)NCC(C(=O)O)c2nccs2)c2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.36
HDAC1 Q13547 2/20 0.36
ALDH1A1 P00352 5/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
SHMT2 P34897 1/20 0.34
POLB P06746 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
RPS6KB1 P23443 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SLC6A9 P48067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982365 0.82 ALDH1A1 (0.34) ALDH1A1LMNASHMT2POLBCYP1A2
SCHEMBL6977286 0.79 ITGB3 (0.53) CYP2C19
SCHEMBL6983774 0.75 ADORA2A (0.40) HDAC3HDAC1SLC6A9
SCHEMBL6985761 0.74 BRD4 (0.37) ALDH1A1LMNAGAAPOLBCYP1A2
Hydrochloric Acid SCHEMBL7346044 0.73 CYP2C19 (0.51) ALDH1A1GAASHMT2POLBCYP1A2
SCHEMBL6980649 0.71 ADORA2A (0.41) GAAPOLBCYP2C19
SCHEMBL6982666 0.70 ADORA2A (0.41) HDAC3HDAC1GAA
SCHEMBL9559011 0.68 ITGB3 (0.63)
SCHEMBL6972650 0.66 ITGB3 (0.38) POLBSLC6A9
SCHEMBL8042923 0.65 ITGB3 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed