SCHEMBL6982539

SCHEMBL6982539

NC(=O)C1=Cn2ccc3cccc(c32)C1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.36
LMNA P02545 1/20 0.32
PIM1 P11309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036977 0.86 MCL1 (0.35)
SCHEMBL6327672 0.81 TRPA1 (0.36) LMNA
SCHEMBL9904854 0.70 LMNA (0.33) LMNA
SCHEMBL3525771 0.67 TRPA1 (0.31) PIM1
SCHEMBL9680591 0.64 TRPA1 (0.32)
SCHEMBL14067698 0.64 NOTUM (0.42) PARP1
SCHEMBL6667856 0.63 TRPA1 (0.36)
SCHEMBL9275405 0.59 PARP1 (0.44) PARP1
SCHEMBL30082247 0.59 PARP1 (0.44) PARP1
SCHEMBL2860722 0.59 MAOA (0.49) PARP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299386-A1 PYRROLOQUINOLONES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-04-09 EP claimed
WO-2002002558-A1 PYRROLOQUINOLONES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-01-10 WO claimed
EP-1299386-A1 PYRROLOQUINOLONES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-04-09 EP disclosed
WO-2002002558-A1 PYRROLOQUINOLONES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-01-10 WO disclosed