SCHEMBL6982789

SCHEMBL6982789

CN1CCC(=O)c2ccn(CCCCCl)c2C1=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.35
ADORA2B P29275 1/20 0.32
POLB P06746 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041754 0.99 PTPN1 (0.34) PTPN1ADORA2BPOLBRECQL
SCHEMBL9041444 0.96 PTPN1 (0.35) PTPN1ADORA2BPOLBRECQL
SCHEMBL6998066 0.92 PTPN1 (0.33) PTPN1ADORA2BPOLBRECQL
SCHEMBL6994882 0.86 PTPN1 (0.31) PTPN1
SCHEMBL9040778 0.86 PTPN1 (0.33) PTPN1ADORA2B
SCHEMBL9040322 0.86 PTPN1 (0.35) PTPN1ADORA2BPOLB
SCHEMBL6989751 0.85 PNMT (0.32) PTPN1
SCHEMBL9041335 0.85 PTPN1 (0.37) PTPN1
SCHEMBL6989876 0.84
SCHEMBL6989871 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0551527-B1 PYRROLOAZEPINE DERIVATIVE SUNTORY LTD (JP) 2003-04-02 EP disclosed
EP-0441349-B1 Pyrroloazepine derivatives SUNTORY LTD (JP) 1996-01-03 EP disclosed
US-5416082-A Antiserotonine agents SUNTORY LIMITED (JP) 1995-05-16 US disclosed
US-5397780-A Antiserotonine, hypotensive, congestive heart failure SUNTORY LIMITED (JP) 1995-03-14 US disclosed
US-5391731-A Useful therapeutics for circulatory diseases SUNTORY LIMITED (JP) 1995-02-21 US disclosed
EP-0551527-A1 PYRROLOAZEPINE DERIVATIVE SUNTORY LIMITED (JP) 1993-07-21 EP disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed