SCHEMBL6983606

SCHEMBL6983606

N=C(N)c1ccc(N(C(=O)CCC(=O)NCC(C(=O)O)n2ccnc2)c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.39
ITGA2B P08514 5/20 0.39
CYP24A1 Q07973 10/20 0.39
CYP27B1 O15528 2/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983967 0.89 ITGB3 (0.51) ITGB3ITGA2BCYP24A1KDM4E
SCHEMBL6981952 0.73 ALDH1A1 (0.49) ITGB3ITGA2BKDM4E
SCHEMBL6984397 0.72 ITGB3 (0.46) ITGB3ITGA2B
SCHEMBL6983016 0.71 ITGB3 (0.47) ITGB3ITGA2BKDM4E
SCHEMBL6981209 0.71 F7 (0.39) ITGB3ITGA2B
SCHEMBL6972650 0.70 ITGB3 (0.38) ITGB3ITGA2B
SCHEMBL9258794 0.69 F2 (0.44) KDM4E
SCHEMBL9558964 0.68 ITGB3 (0.69) ITGB3ITGA2B
SCHEMBL6985725 0.68 ITGB3 (0.43) ITGB3ITGA2B
SCHEMBL9426106 0.67 ITGB3 (0.48) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630366-B1 SUBSTITUTED HETEROCYCLIC DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 2003-01-02 EP disclosed
EP-0539343-B1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO CO (US) 2000-07-26 EP disclosed
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed