SCHEMBL6984197

SCHEMBL6984197

CC(C)N1Cc2cc(C(N)=O)ccc2N(CCCl)S1(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HSD17B3 P37058 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC3 O15379 1/20 0.36
CYP2C19 P33261 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
OPRM1 P35372 4/20 0.35
OPRK1 P41145 4/20 0.35
OPRD1 P41143 3/20 0.34
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985472 0.90 MAPT (0.38) ALDH1A1KMT2A
SCHEMBL6975363 0.87 SRD5A1 (0.41) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL8318057 0.79 KDM4E (0.39) KDM4EOPRM1RORC
SCHEMBL6984303 0.77 BRD4 (0.32) ALDH1A1MEN1KMT2ABRD4RORC
SCHEMBL8316061 0.74 CRY1 (0.35)
SCHEMBL8317987 0.70 ADRA2A (0.36) KDM4EALDH1A1HSD17B3RORC
SCHEMBL26075696 0.64 HSD17B3 (0.52) KDM4EALDH1A1HSD17B10HSD17B3SIRT2
SCHEMBL7089097 0.62 BMPR1B (0.45) KDM4EALDH1A1HSD17B10HSD17B3SIRT2
SCHEMBL30197112 0.61 ALDH1A1 (0.53) KDM4EALDH1A1HSD17B10SIRT2HDAC1
SCHEMBL12199408 0.61 ALDH1A1 (0.55) KDM4EALDH1A1HSD17B10HSD17B3SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131321-B1 INDOLE DERIVATIVES AND THEIR USE AS SEROTONIN RECEPTOR LIGANDS LILLY CO ELI (GB) 2003-09-10 EP disclosed
US-6329366-B1 HETEROCYCLIC, PIPERIDINE, INDOLE DERIVITIVES FOR TREATMENT OF NERVOUS SYSTEM DISORDERS AND SEROTONIN ANTAGONIST ELI LILLY AND COMPANY LIMITED (GB) 2001-12-11 US disclosed