SCHEMBL6985472

SCHEMBL6985472

CC(=O)c1ccc2c(c1)CN(C(C)C)S(=O)(=O)N2CCCl

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
KCNJ1 P48048 2/20 0.34
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
HSD17B1 P14061 1/20 0.32
KMT2A Q03164 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ACACB O00763 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984197 0.90 KDM4E (0.41) KMT2AALDH1A1
SCHEMBL6975363 0.88 SRD5A1 (0.41) MAPTNPC1MAPK1KMT2AALDH1A1
SCHEMBL6984303 0.78 BRD4 (0.32) KMT2AALDH1A1
SCHEMBL8316061 0.75 CRY1 (0.35)
SCHEMBL8317987 0.71 ADRA2A (0.36) PKML3MBTL1ALDH1A1ACACB
SCHEMBL6978812 0.68 MAPT (0.40) MAPTHPGDNPC1RAB9AKCNJ1
SCHEMBL18876729 0.63 NPC1 (0.58) MAPTHPGDNPC1RAB9AKCNJ1
SCHEMBL4889668 0.61 MCHR1 (0.36) MAPTHPGDRAB9AL3MBTL1ALDH1A1
SCHEMBL3230153 0.60 POLB (0.46) MAPTHPGDKMT2AALDH1A1
SCHEMBL937684 0.60 MAPT (0.55) MAPTHPGDNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131321-B1 INDOLE DERIVATIVES AND THEIR USE AS SEROTONIN RECEPTOR LIGANDS LILLY CO ELI (GB) 2003-09-10 EP disclosed
US-6329366-B1 HETEROCYCLIC, PIPERIDINE, INDOLE DERIVITIVES FOR TREATMENT OF NERVOUS SYSTEM DISORDERS AND SEROTONIN ANTAGONIST ELI LILLY AND COMPANY LIMITED (GB) 2001-12-11 US disclosed