SCHEMBL6984288

SCHEMBL6984288

N=C(NC(=O)OCc1ccccc1)c1ccc(CCC(=O)N2CCCc3cc(N(CCN4CCOCC4)S(=O)(=O)c4cccc5ccccc45)ccc32)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 5/20 0.35
ALDH1A1 P00352 3/20 0.34
CASR P41180 1/20 0.34
RORC P51449 1/20 0.34
F10 P00742 1/20 0.33
F7 P08709 1/20 0.33
EPHX2 P34913 2/20 0.32
PARP1 P09874 1/20 0.32
TP53 P04637 1/20 0.31
AURKA O14965 1/20 0.31
FLT1 P17948 1/20 0.31
KDR P35968 1/20 0.31
FLT3 P36888 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085092 0.90 ALDH1A1 (0.39) NR3C1ALDH1A1RORCPARP1TP53
Hydrochloric Acid SCHEMBL7086319 0.87 F10 (0.42) NR3C1ALDH1A1RORCF10F7
SCHEMBL7088163 0.87 PARP1 (0.37) NR3C1ALDH1A1PARP1TP53
SCHEMBL7089638 0.86 PARP1 (0.36) NR3C1ALDH1A1RORCPARP1TP53
SCHEMBL6984290 0.85 F10 (0.35) NR3C1ALDH1A1CASRRORCF10
SCHEMBL6978633 0.82 RORC (0.36) NR3C1ALDH1A1RORCPARP1TP53
SCHEMBL6981576 0.81 NR3C1 (0.44) NR3C1
SCHEMBL7084262 0.77 F2 (0.46) NR3C1ALDH1A1RORCF10F7
SCHEMBL6981981 0.76 F2 (0.40) NR3C1ALDH1A1RORCF10F7
SCHEMBL6978671 0.76 F2 (0.46) NR3C1ALDH1A1RORCF10PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed