SCHEMBL6984337

SCHEMBL6984337

CCCCOC(=O)N1CCN(c2nccc(C(=O)O)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ACHE P22303 2/20 0.44
HRH2 P25021 2/20 0.43
HRH1 P35367 2/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTPN11 Q06124 1/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
ATM Q13315 1/20 0.42
P2RY12 Q9H244 7/20 0.42
HTT P42858 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
SMYD3 Q9H7B4 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136906 0.79 ACHE (0.63) ACHEPOLBPTPN11MAPT
SCHEMBL6986404 0.79 POLB (0.48) MEN1KMT2AHRH2HRH1LMNA
SCHEMBL31705889 0.78 ACHE (0.57) MEN1KMT2AACHEPTPN11ALDH1A1
SCHEMBL31635767 0.76 TRPV1 (0.51) HRH2HRH1LMNAPOLBSMN1; SMN2
SCHEMBL7243129 0.75 KMT2A (0.53) MEN1KMT2AHRH2HRH1LMNA
SCHEMBL15188017 0.75 ACHE (0.49) ACHEHTT
SCHEMBL27470853 0.74 HRH4 (0.53) MEN1KMT2APOLBOPRD1OPRK1
SCHEMBL1459682 0.74 MAPT (0.57) MEN1KMT2AHRH2HRH1LMNA
SCHEMBL28070878 0.73 MAPK8 (0.52) ACHEPOLBSMN1; SMN2PTPN11ALDH1A1
SCHEMBL9405372 0.72 POLB (0.73) HRH2HRH1LMNAPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed